Eugenio Uriarte Villares
AuthID: R-001-GGC
41
TITLE: New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies Full Text
AUTHORS: Francesca Pintus; Maria J Matos ; Santiago Vilar; George Hripcsak; Carla Varela; Eugenio Uriarte; Lourdes Santana; Fernanda Borges ; Rosaria Medda; Amalia Di Petrillo; Benedetta Era; Antonella Fais;
PUBLISHED: 2017, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 25, ISSUE: 5
AUTHORS: Francesca Pintus; Maria J Matos ; Santiago Vilar; George Hripcsak; Carla Varela; Eugenio Uriarte; Lourdes Santana; Fernanda Borges ; Rosaria Medda; Amalia Di Petrillo; Benedetta Era; Antonella Fais;
PUBLISHED: 2017, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 25, ISSUE: 5
42
TITLE: Coumarin versus Chromone Monoamine Oxidase B Inhibitors: Quo Vadis? Full Text
AUTHORS: Andre Fonseca; Joana Reis; Tiago Silva; Maria Joao Matos ; Donatella Bagetta; Francesco Ortuso; Stefano Alcaro; Eugenio Uriarte; Fernanda Borges ;
PUBLISHED: 2017, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 60, ISSUE: 16
AUTHORS: Andre Fonseca; Joana Reis; Tiago Silva; Maria Joao Matos ; Donatella Bagetta; Francesco Ortuso; Stefano Alcaro; Eugenio Uriarte; Fernanda Borges ;
PUBLISHED: 2017, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 60, ISSUE: 16
43
TITLE: In silico genotoxicity of coumarins: Application of the Phenol-Explorer food database to functional food science
AUTHORS: Guardado Yordi, E; Matos, MJ ; Pérez Martínez, A; Tornes, AC; Santana, L; Molina, E; Uriarte, E;
PUBLISHED: 2017, SOURCE: Food and Function, VOLUME: 8, ISSUE: 8
AUTHORS: Guardado Yordi, E; Matos, MJ ; Pérez Martínez, A; Tornes, AC; Santana, L; Molina, E; Uriarte, E;
PUBLISHED: 2017, SOURCE: Food and Function, VOLUME: 8, ISSUE: 8
44
TITLE: Synthesis and structure-activity relationship study of novel 3-heteroarylcoumarins based on pyridazine scaffold as selective MAO-B inhibitors Full Text
AUTHORS: Costas Lago, MC; Besada, P; Rodriguez Enriquez, F; Vina, D; Vilar, S; Uriarte, E; Borges, F ; Teran, C;
PUBLISHED: 2017, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 139
AUTHORS: Costas Lago, MC; Besada, P; Rodriguez Enriquez, F; Vina, D; Vilar, S; Uriarte, E; Borges, F ; Teran, C;
PUBLISHED: 2017, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 139
INDEXED IN: Scopus WOS
45
TITLE: Synthesis and structure-activity relationship study of novel 3-heteroarylcoumarins based on pyridazine scaffold as selective MAO-B inhibitors Full Text
AUTHORS: María Carmen Costas-Lago; Pedro Besada; Fernanda Rodríguez-Enríquez; Dolores Viña; Santiago Vilar; Eugenio Uriarte; Fernanda Borges ; Carmen Terán;
PUBLISHED: 2017, SOURCE: European Journal of Medicinal Chemistry, VOLUME: 139
AUTHORS: María Carmen Costas-Lago; Pedro Besada; Fernanda Rodríguez-Enríquez; Dolores Viña; Santiago Vilar; Eugenio Uriarte; Fernanda Borges ; Carmen Terán;
PUBLISHED: 2017, SOURCE: European Journal of Medicinal Chemistry, VOLUME: 139
46
TITLE: Progress in the development of small molecules as new human A(3) adenosine receptor ligands based on the 3-thiophenylcoumarin core
AUTHORS: Matos, MJ ; Vilar, S; Kachler, S; Vazquez Rodriguez, S; Varela, C; Delogu, G; Hripcsak, G; Santana, L; Uriarte, E; N Klotz; Borges, F ;
PUBLISHED: 2016, SOURCE: MEDCHEMCOMM, VOLUME: 7, ISSUE: 5
AUTHORS: Matos, MJ ; Vilar, S; Kachler, S; Vazquez Rodriguez, S; Varela, C; Delogu, G; Hripcsak, G; Santana, L; Uriarte, E; N Klotz; Borges, F ;
PUBLISHED: 2016, SOURCE: MEDCHEMCOMM, VOLUME: 7, ISSUE: 5
47
TITLE: Exploring coumarin potentialities: development of new enzymatic inhibitors based on the 6-methyl-3-carboxamidocoumarin scaffold
AUTHORS: Fonseca, A; Matos, MJ ; Reis, J; Duarte, Y; Gutierrez, M; Santana, L; Uriarte, E; Borges, F ;
PUBLISHED: 2016, SOURCE: RSC ADVANCES, VOLUME: 6, ISSUE: 55
AUTHORS: Fonseca, A; Matos, MJ ; Reis, J; Duarte, Y; Gutierrez, M; Santana, L; Uriarte, E; Borges, F ;
PUBLISHED: 2016, SOURCE: RSC ADVANCES, VOLUME: 6, ISSUE: 55
48
TITLE: Discovery of New Chemical Entities for Old Targets: Insights on the Lead Optimization of Chromone-Based Monoamine Oxidase B (MAO-B) Inhibitors Full Text
AUTHORS: Joana Reis; Fernando Cagide ; Daniel Chavarria ; Tiago Silva; Carlos Fernandes; Alexandra Gaspar ; Eugenio Uriarte; Fernando Remiao ; Stefano Alcaro; Francesco Ortuso; Fernanda Borges ;
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 12
AUTHORS: Joana Reis; Fernando Cagide ; Daniel Chavarria ; Tiago Silva; Carlos Fernandes; Alexandra Gaspar ; Eugenio Uriarte; Fernando Remiao ; Stefano Alcaro; Francesco Ortuso; Fernanda Borges ;
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 12
49
TITLE: Development of Blood-Brain Barrier Permeable Nitrocatechol-Based Catechol O-Methyltransferase Inhibitors with Reduced Potential for Hepatotoxicity Full Text
AUTHORS: Tiago Silva; Tarek Mohamed; Arash Shakeri; Praveen P N Rao; Loreto Martinez Gonzalez; Daniel I Perez; Ana Martinez; Maria Joao Valente; Jorge Garrido; Eugenio Uriarte; Paula Serrao ; Patricio Soares da Silva; Fernando Remiao ; Fernanda Borges ;
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
AUTHORS: Tiago Silva; Tarek Mohamed; Arash Shakeri; Praveen P N Rao; Loreto Martinez Gonzalez; Daniel I Perez; Ana Martinez; Maria Joao Valente; Jorge Garrido; Eugenio Uriarte; Paula Serrao ; Patricio Soares da Silva; Fernando Remiao ; Fernanda Borges ;
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
50
TITLE: Computational Drug Target Screening through Protein Interaction Profiles Full Text
AUTHORS: Santiago Vilar; Elias Quezada; Eugenio Uriarte; Stefano Costanzi; Fernanda Borges ; Dolores Vina; George Hripcsak;
PUBLISHED: 2016, SOURCE: SCIENTIFIC REPORTS, VOLUME: 6, ISSUE: 1
AUTHORS: Santiago Vilar; Elias Quezada; Eugenio Uriarte; Stefano Costanzi; Fernanda Borges ; Dolores Vina; George Hripcsak;
PUBLISHED: 2016, SOURCE: SCIENTIFIC REPORTS, VOLUME: 6, ISSUE: 1