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TITLE: Selective Inhibition of Bruton?s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
AUTHORS: Sousa, Barbara B.; De Almeida, Catia Rebelo; Barahona, Ana F.; Lopes, Raquel; Martins Logrado, Ana; Cavaco, Marco; Neves, Vera; Carvalho, Luis A. R.; Labao Almeida, Carlos; Coelho, Ana R.; Bento, Marta Leal; Lopes, Ricardo M. R. M.; Oliveira, Bruno L.; Castanho, Miguel A. R. B.; Neumeister, Peter; Deutsch, Alexander; Vladimer, Gregory I.; Krall, Nikolaus; Joao, Cristina; Corzana, Francisco; Seixas, Joao D.; Fior, Rita; Bernardes, Goncalo J. L.; ...More
PUBLISHED: 2022, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 5, ISSUE: 11

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TITLE: Facile installation of post-translational modifications on the tau protein via chemical mutagenesis
AUTHORS: Vendruscolo, M; Bernardes, GJL; Lindstedt, PR; Taylor, RJ;
PUBLISHED: 2021, SOURCE: ACS Chemical Neuroscience

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TITLE: Facile Installation of Post-translational Modifications on the Tau Protein via Chemical Mutagenesis
AUTHORS: Lindstedt, PR; Taylor, RJ; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 3

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TITLE: Precise protein conjugation technology for the construction of homogenous glycovaccines
AUTHORS: Kitowski, A; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: Drug Discovery Today: Technologies

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Scopus

TITLE: The role of reversible and irreversible covalent chemistry in targeted protein degradation
AUTHORS: Kiely Collins, H; Winter, GE; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 28, ISSUE: 7

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TITLE: Exploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation Full Text
AUTHORS: Neukirch, K; Alsabil, K; Dinh, CP; Bilancia, R; Raasch, M; Ville, A; Cerqua, I; Viault, G; Breard, D; Pace, S; Temml, V; Brunner, E; Jordan, PM; Marques, MC; Loeser, K; Gollowitzer, A; Permann, S; Gerstmeier, J; Lorkowski, S; Stuppner, H; Garscha, U; Rodrigues, T; Bernardes, GJL; Schuster, D; Seraphin, D; Richomme, P; Rossi, A; Mosig, AS; Roviezzo, F; Werz, O; Helesbeux, JJ; Koeberle, A; ...More
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15

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TITLE: Dichloro Butenediamides as Irreversible Site-Selective Protein Conjugation Reagent Full Text
AUTHORS: Laserna, V; Abegg, D; Afonso, CF; Martin, EM; Adibekian, A; Ravn, P; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

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TITLE: Combating small-molecule aggregation with machine learning
AUTHORS: Lee, K; Yang, A; Lin, YC; Reker, D; Bernardes, GJL; Rodrigues, T;
PUBLISHED: 2021, SOURCE: CELL REPORTS PHYSICAL SCIENCE, VOLUME: 2, ISSUE: 9

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TITLE: A Platform for Site-Specific DNA-Antibody Bioconjugation by Using Benzoylacrylic-Labelled Oligonucleotides Full Text
AUTHORS: Konc, J; Brown, L; Whiten, DR; Zuo, YK; Ravn, P; Klenerman, D; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

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TITLE: Diazaborines Are a Versatile Platform to Develop ROS-Responsive Antibody Drug Conjugates** Full Text
AUTHORS: Antonio, JPM; Carvalho, JI; Andre, AS; Dias, JNR; Aguiar, SI; Faustino, H; Lopes, RMRM; Veiros, LF; Bernardes, GJL; Silva, FA; Gois, PMP;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

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