Jorge António Ribeiro Salvador
AuthID: R-000-7NJ
31
TITLE: Chalcone derivatives targeting mitosis: synthesis, evaluation of antitumor activity and lipophilicity Full Text
AUTHORS: Patricia Pinto; Carmen Mariana Machado; Joana Moreira; Jose Diogo P Almeida; Patricia M A Silva; Ana C Henriques; Jose X Soares ; Jorge A R Salvador; Carlos Afonso ; Madalena Pinto; Hassan Bousbaa; Honorina Cidade ;
PUBLISHED: 2019, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 184
AUTHORS: Patricia Pinto; Carmen Mariana Machado; Joana Moreira; Jose Diogo P Almeida; Patricia M A Silva; Ana C Henriques; Jose X Soares ; Jorge A R Salvador; Carlos Afonso ; Madalena Pinto; Hassan Bousbaa; Honorina Cidade ;
PUBLISHED: 2019, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 184
32
TITLE: Structural insights and binding analysis for determining the molecular bases for programmed cell death protein ligand-1 inhibition
AUTHORS: Acúrcio, RC; Leonardo Sousa, C; García Sosa, AT; Salvador, JA; Florindo, HF; Guedes, RC;
PUBLISHED: 2019, SOURCE: MedChemComm, VOLUME: 10, ISSUE: 10
AUTHORS: Acúrcio, RC; Leonardo Sousa, C; García Sosa, AT; Salvador, JA; Florindo, HF; Guedes, RC;
PUBLISHED: 2019, SOURCE: MedChemComm, VOLUME: 10, ISSUE: 10
33
TITLE: Chemical Patterns of Proteasome Inhibitors: Lessons Learned from Two Decades of Drug Design
AUTHORS: Guedes, RA; Aniceto, N; Andrade, MAP; Salvador, JAR; Guedes, RC;
PUBLISHED: 2019, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 20, ISSUE: 21
AUTHORS: Guedes, RA; Aniceto, N; Andrade, MAP; Salvador, JAR; Guedes, RC;
PUBLISHED: 2019, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 20, ISSUE: 21
34
TITLE: An overview of glutaminyl cyclase inhibitors for Alzheimer's disease
AUTHORS: Coimbra, JRM; Sobral, PJM; Santos, AE; Moreira, PI; Moreira, Paula Isabel; Paula I. Moreira ; Salvador, JAR;
PUBLISHED: 2019, SOURCE: FUTURE MEDICINAL CHEMISTRY, VOLUME: 11, ISSUE: 24
AUTHORS: Coimbra, JRM; Sobral, PJM; Santos, AE; Moreira, PI; Moreira, Paula Isabel; Paula I. Moreira ; Salvador, JAR;
PUBLISHED: 2019, SOURCE: FUTURE MEDICINAL CHEMISTRY, VOLUME: 11, ISSUE: 24
35
TITLE: Synthesis and Biological Evaluation of New Madecassic Acid Derivatives Targeting ERK Cascade Signaling
AUTHORS: Valdeira, ASC; Ritt, DA; Morrison, DK; McMahon, JB; Gustafson, KR; Salvador, JAR;
PUBLISHED: 2018, SOURCE: FRONTIERS IN CHEMISTRY, VOLUME: 6
AUTHORS: Valdeira, ASC; Ritt, DA; Morrison, DK; McMahon, JB; Gustafson, KR; Salvador, JAR;
PUBLISHED: 2018, SOURCE: FRONTIERS IN CHEMISTRY, VOLUME: 6
36
TITLE: Structure-Function Analysis of Immune Checkpoint Receptors to Guide Emerging Anticancer Immunotherapy
AUTHORS: Acurcio, RC; Scomparin, A; Conniot, J; Salvador, JAR; Satchi Fainaro, R; Florindo, HF; Guedes, RC;
PUBLISHED: 2018, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 61, ISSUE: 24
AUTHORS: Acurcio, RC; Scomparin, A; Conniot, J; Salvador, JAR; Satchi Fainaro, R; Florindo, HF; Guedes, RC;
PUBLISHED: 2018, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 61, ISSUE: 24
37
TITLE: Highlights in BACE1 inhibitors for Alzheimer's disease treatment
AUTHORS: Judite R M Coimbra; Daniela F F Marques; Salete J Baptista; Cláudia M F Pereira; Paula I Moreira; Teresa C P Dinis; Armanda E Santos; Jorge A R Salvador;
PUBLISHED: 2018, SOURCE: Frontiers in Chemistry, VOLUME: 6, ISSUE: MAY
AUTHORS: Judite R M Coimbra; Daniela F F Marques; Salete J Baptista; Cláudia M F Pereira; Paula I Moreira; Teresa C P Dinis; Armanda E Santos; Jorge A R Salvador;
PUBLISHED: 2018, SOURCE: Frontiers in Chemistry, VOLUME: 6, ISSUE: MAY
38
TITLE: Novel PARP-1 Inhibitor Scaffolds Disclosed by a Dynamic Structure-Based Pharmacophore Approach
AUTHORS: Baptista, SJ; Silva, MMC; Moroni, E; Meli, M; Colombo, G; Dinis, TCP; Salvador, JAR;
PUBLISHED: 2017, SOURCE: PLOS ONE, VOLUME: 12, ISSUE: 1
AUTHORS: Baptista, SJ; Silva, MMC; Moroni, E; Meli, M; Colombo, G; Dinis, TCP; Salvador, JAR;
PUBLISHED: 2017, SOURCE: PLOS ONE, VOLUME: 12, ISSUE: 1
39
TITLE: Design, synthesis and biological evaluation of novel C-29 carbamate celastrol derivatives as potent and selective cytotoxic compounds
AUTHORS: Figueiredo, SAC; Salvador, JAR; Cortés, R; Cascante, M;
PUBLISHED: 2017, SOURCE: European Journal of Medicinal Chemistry, VOLUME: 139
AUTHORS: Figueiredo, SAC; Salvador, JAR; Cortés, R; Cascante, M;
PUBLISHED: 2017, SOURCE: European Journal of Medicinal Chemistry, VOLUME: 139
40
TITLE: Novel celastrol derivatives with improved selectivity and enhanced antitumour activity: Design, synthesis and biological evaluation
AUTHORS: Figueiredo, SAC; Salvador, JAR; Cortes, R; Cascante, M;
PUBLISHED: 2017, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 138
AUTHORS: Figueiredo, SAC; Salvador, JAR; Cortes, R; Cascante, M;
PUBLISHED: 2017, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 138