Rui Ferreira Alves Moreira
AuthID: R-000-FTJ
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TITLE: Structural Optimization of Antimycobacterial Azaaurones Towards Improved Solubility and Metabolic Stability Full Text
AUTHORS: André Campaniço; Shrika Harjivan; Elisabete Freitas; Marco Serafini; Manuela Gaspar; Rita Capela; Pedro Gomes; Audrey Jordaan; Ana Madureira; Vânia André; Andreia Silva; Teresa Duarte; Isabel Portugal; João Perdigão; Rui Moreira; Digby Warner; Francisca Lopes;
PUBLISHED: 2023, SOURCE: ChemMedChem, VOLUME: 18, ISSUE: 24
AUTHORS: André Campaniço; Shrika Harjivan; Elisabete Freitas; Marco Serafini; Manuela Gaspar; Rita Capela; Pedro Gomes; Audrey Jordaan; Ana Madureira; Vânia André; Andreia Silva; Teresa Duarte; Isabel Portugal; João Perdigão; Rui Moreira; Digby Warner; Francisca Lopes;
PUBLISHED: 2023, SOURCE: ChemMedChem, VOLUME: 18, ISSUE: 24
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TITLE: New azaaurone derivatives as potential multitarget agents in HIV-TB coinfection Full Text
AUTHORS: Leite, Debora I.; Campanico, Andre; Costa, Pedro A. G.; Correa, Isadora A.; da Costa, Luciana J.; Bastos, Monica M.; Moreira, Rui; Lopes, Francisca; Jordaan, Audrey; Warner, Digby F.; Boechat, Nubia;
PUBLISHED: 2023, SOURCE: ARCHIV DER PHARMAZIE, VOLUME: 357, ISSUE: 2
AUTHORS: Leite, Debora I.; Campanico, Andre; Costa, Pedro A. G.; Correa, Isadora A.; da Costa, Luciana J.; Bastos, Monica M.; Moreira, Rui; Lopes, Francisca; Jordaan, Audrey; Warner, Digby F.; Boechat, Nubia;
PUBLISHED: 2023, SOURCE: ARCHIV DER PHARMAZIE, VOLUME: 357, ISSUE: 2
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TITLE: New Compound Combining an Integrase-Targeting Aptamer and a Small Interfering RNA Targeting the Trans-Activation Response/Poly A Region of HIV-1 Potently Suppresses HIV-1 Replication
AUTHORS: Inês Moranguinho; Pedro Borrego; João Lavrado; Rui Moreira; Nuno Taveira;
PUBLISHED: 2023, SOURCE: The 6th International Congress of CiiEM—Immediate and Future Challenges to Foster One Health
AUTHORS: Inês Moranguinho; Pedro Borrego; João Lavrado; Rui Moreira; Nuno Taveira;
PUBLISHED: 2023, SOURCE: The 6th International Congress of CiiEM—Immediate and Future Challenges to Foster One Health
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TITLE: Tandem Thio-Michael Addition/Remote Lactone Activation of 5-Hydroxymethylfurfural-Derived delta-Lactone-Fused Cyclopentenones Full Text
AUTHORS: Gomes, RFA; Ravasco, JMJM; Andrade, KHS; Coelho, JAS; Moreira, R; Oliveira, R; Nogueira, F; Afonso, CAM;
PUBLISHED: 2022, SOURCE: CHEMSUSCHEM, VOLUME: 15, ISSUE: 13
AUTHORS: Gomes, RFA; Ravasco, JMJM; Andrade, KHS; Coelho, JAS; Moreira, R; Oliveira, R; Nogueira, F; Afonso, CAM;
PUBLISHED: 2022, SOURCE: CHEMSUSCHEM, VOLUME: 15, ISSUE: 13
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TITLE: Indole-Containing Pyrazino[2,1-b]quinazoline-3,6-diones Active against Plasmodium and Trypanosomatids
AUTHORS: Long, S; Duarte, D; Carvalho, C; Oliveira, R; Santarem, N; Palmeira, A ; Resende, DISP; Silva, AMS; Moreira, R; Kijjoa, A; da Silva, AC ; Nogueira, F; Sousa, E ; Pinto, MMM;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 2
AUTHORS: Long, S; Duarte, D; Carvalho, C; Oliveira, R; Santarem, N; Palmeira, A ; Resende, DISP; Silva, AMS; Moreira, R; Kijjoa, A; da Silva, AC ; Nogueira, F; Sousa, E ; Pinto, MMM;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 2
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TITLE: Inflammatory biomarkers in staging of chronic kidney disease: elevated TNFR2 levels accompanies renal function decline Full Text
AUTHORS: Lousa, Irina; Belo, Luis ; Valente, Maria Joao; Rocha, Susana; Preguica, Ines; Rocha Pereira, Petronila; Beirao, Idalina; Mira, Filipe; Alves, Rui; Reis, Flavio; Alice Santos-Silva ;
PUBLISHED: 2022, SOURCE: INFLAMMATION RESEARCH, VOLUME: 71, ISSUE: 5-6
AUTHORS: Lousa, Irina; Belo, Luis ; Valente, Maria Joao; Rocha, Susana; Preguica, Ines; Rocha Pereira, Petronila; Beirao, Idalina; Mira, Filipe; Alves, Rui; Reis, Flavio; Alice Santos-Silva ;
PUBLISHED: 2022, SOURCE: INFLAMMATION RESEARCH, VOLUME: 71, ISSUE: 5-6
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TITLE: Harnessing Protein-Ligand Interaction Fingerprints to Predict New Scaffolds of RIPK1 Inhibitors Full Text
AUTHORS: Aniceto, Natalia; Marques, Vanda; Amaral, Joana D.; Serra, Patricia A.; Moreira, Rui; Rodrigues, Cecilia M. P.; Guedes, Rita C.;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 15
AUTHORS: Aniceto, Natalia; Marques, Vanda; Amaral, Joana D.; Serra, Patricia A.; Moreira, Rui; Rodrigues, Cecilia M. P.; Guedes, Rita C.;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 15
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TITLE: Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Orally Bioavailable, and Blood-Brain Barrier Penetrant PROTAC Degrader of Leucine-Rich Repeat Kinase 2
AUTHORS: Liu, Xingui; Kalogeropulou, Alexia F.; Domingos, Sofia; Makukhin, Nikolai; Nirujogi, Raja S.; Singh, Francois; Shpiro, Natalia; Saalfrank, Anton; Sammler, Esther; Ganley, Ian G.; Moreira, Rui; Alessi, Dario R.; Ciulli, Alessio;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 37
AUTHORS: Liu, Xingui; Kalogeropulou, Alexia F.; Domingos, Sofia; Makukhin, Nikolai; Nirujogi, Raja S.; Singh, Francois; Shpiro, Natalia; Saalfrank, Anton; Sammler, Esther; Ganley, Ian G.; Moreira, Rui; Alessi, Dario R.; Ciulli, Alessio;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 37
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TITLE: Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 61, ISSUE: 47
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 61, ISSUE: 47
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TITLE: The Facets of Diversity: The EFMC Perspective
AUTHORS: Borsari, Chiara; Matagne, Brieuc; Goncharenko, Kristina; Moreira, Rui; Auberson, Yves P.;
PUBLISHED: 2022, SOURCE: CHEMMEDCHEM, VOLUME: 18, ISSUE: 1
AUTHORS: Borsari, Chiara; Matagne, Brieuc; Goncharenko, Kristina; Moreira, Rui; Auberson, Yves P.;
PUBLISHED: 2022, SOURCE: CHEMMEDCHEM, VOLUME: 18, ISSUE: 1