51
TITLE: VScore: uma plataforma para desenvolvimento de novos fármacos usando screening virtual
AUTHORS: Hugo J Froufe; Isabel C Ferreira; João N Sousa; José Rufino; Rui M Abreu;
PUBLISHED: 2013, SOURCE: V Workshop em Bioinformática. Escola Superior Agrária de Bragança, 15 e 16 de Maio de 2013
INDEXED IN: Handle
52
TITLE: Evaluation of growth inhibitory activity of Crataegus monogyna Jacq. flower bud extracts against human tumor cell lines
AUTHORS: João C Barreira; Rui M Abreu; Sandra Rodrigues; Ana M Carvalho; Isabel C Ferreira;
PUBLISHED: 2013, SOURCE: 1st Symposium on Medicinal Chemistry of University of Minho. 17 de Maio de 2013
INDEXED IN: Handle
53
TITLE: Virtual screening of thieno[3,2-b]pyridine arylthioether (hetero)aryltriazole derivatives as potential tyrosine kinase VEGFR2 inhibitors.
AUTHORS: Ricardo C Calhelha; Agathe Begouin; Joana F Campos; Isabel C Ferreira; Maria J R Queiroz; Rui M Abreu;
PUBLISHED: 2013, SOURCE: XIX Encontro Galego-Português de Química
INDEXED IN: Handle
54
TITLE: New di(heteroaryl)thioethers 1,3-diarylureas in the thieno[3,2-b]pyridine series as VEGFR2 tyrosine kinase inhibitors: docking, synthesis, enzymatic and cellular assays
AUTHORS: Vera A Machado; Raquel Costa; Daniela Peixoto; Rui M Abreu; Ricardo C Calhelha; Isabel C Ferreira; Raquel Soares; Maria J R Queiroz;
PUBLISHED: 2013, SOURCE: 49th International Conference on Medicinal Chemistry (RICT 2013)
INDEXED IN: Handle
55
TITLE: Synthesis and evaluation of the antitumor potential of new aminated or methoxylated di(hetero)arylthioethers in the thieno[3,2-b]pyridine series
AUTHORS: Ricardo C Calhelha; Joana F Campos; Daniela Peixoto; Rui M Abreu; Isabel C Ferreira; Maria J R Queiroz;
PUBLISHED: 2013, SOURCE: 1st Symposium on Medicinal Chemistry of University of Minho
INDEXED IN: Handle
56
TITLE: Synthesis of new N-[3-(thieno[3,2-b]pyridine-7-ylthio)phenyl]benzamides as potential inhibitors the tyrosine kinase domain of VEGFR2
AUTHORS: Joana F Campos; Agathe Begouin; Daniela Peixoto; Hugo J Froufe; Rui M Abreu; Isabel C Ferreira; Maria J R Queiroz;
PUBLISHED: 2013, SOURCE: 1st Symposium on Medicinal Chemistry of University of Minho
INDEXED IN: Handle
57
TITLE: Epidermal growth factor receptor inhibitory activity of new potential antitumor di(hetero)arylethers and di(hetero)arylamines in the thieno[3,2-b]pyridine series
AUTHORS: Ricardo C Calhelha; Daniela Peixoto; Pedro Soares; Isabel C Ferreira; Rui M Abreu; Maria J R Queiroz;
PUBLISHED: 2013, SOURCE: 1st International Symposium on Profiling
INDEXED IN: Handle
58
TITLE: Synthesis, growth inhibitory activity on human tumor cell lines and evaluation of the hepatotoxicity of di(hetero)arylethers and di(hetero)arylamines in the thieno[3,2-b]pyridine series.
AUTHORS: Ricardo C Calhelha; Daniela Peixoto; Pedro Soares; Isabel C Ferreira; Rui M Abreu; Maria J R Queiroz;
PUBLISHED: 2012, SOURCE: 3º Encontro Nacional de Química Terapêutica e 1st Portuguese-Spanish-Brazilian Meeting on Medicinal Chemistry, 28 a 30 de Novembro
INDEXED IN: Handle
59
TITLE: Heteroarylether 1,3-diarylureas in the thieno[3,2-d]pyrimidine series as VEGFR2 tyrosine Kinase inhibitors: synthesis, docking studies, enzymatic and cellular assays
AUTHORS: Maria J R Queiroz; Daniela Peixoto; Pedro Soares; Rui M Abreu; Hugo J Froufe; Ricardo C Calhelha; Isabel C Ferreira; Raquel Costa; Raquel Soares;
PUBLISHED: 2012, SOURCE: 48th International conference on Medicinal Chemistry. Interfacing Chemical Biology and Drug Discovery, 4-6 July 2012.
INDEXED IN: Handle
60
TITLE: Synthesis of novel 1-aryl-3-[2,3- or 4-(thieno[3,2-b]pyridin-7-ylthio)phenyl]ureas and evaluation as VEGFR2 tyrosine kinase inhibitors
AUTHORS: Daniela Peixoto; Maria J R Queiroz; Rui M Abreu; Hugo J Froufe; Ricardo C Calhelha; Isabel C Ferreira;
PUBLISHED: 2012, SOURCE: XXIInd International Symposium on Medicinal Chemistry, 2-6th September 2012
INDEXED IN: Handle
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