Giacomo Landi
AuthID: R-00G-YQF
1
TITLE: The discovery of aryl-2-nitroethyl triamino pyrimidines as <i>anti-Trypanosoma brucei</i> agents Full Text
AUTHORS: Linciano, Pasquale; Pozzi, Cecilia; Tassone, Giusy; Landi, Giacomo; Mangani, Stefano; Santucci, Matteo; Luciani, Rosaria; Ferrari, Stefania; Santarem, Nuno; Tagliazucchi, Lorenzo; Cordeiro da Silva, Anabela; Tonelli, Michele; Tondi, Donatella; Bertarini, Laura; Gul, Sheraz; Witt, Gesa; Moraes, Carolina B.; Costantino, Luca; Costi, Maria Paola;
PUBLISHED: 2024, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 264
AUTHORS: Linciano, Pasquale; Pozzi, Cecilia; Tassone, Giusy; Landi, Giacomo; Mangani, Stefano; Santucci, Matteo; Luciani, Rosaria; Ferrari, Stefania; Santarem, Nuno; Tagliazucchi, Lorenzo; Cordeiro da Silva, Anabela; Tonelli, Michele; Tondi, Donatella; Bertarini, Laura; Gul, Sheraz; Witt, Gesa; Moraes, Carolina B.; Costantino, Luca; Costi, Maria Paola;
PUBLISHED: 2024, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 264
INDEXED IN: 
Scopus 
WOS
Scopus WOS2
TITLE: Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents
AUTHORS: Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Simo, Claude U. Konchie; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarem, Nuno; Tavares, Joana; Cordeiro da Silva, Anabela; Costi, Maria Paola; Tonelli, Michele;
PUBLISHED: 2024, SOURCE: ACS INFECTIOUS DISEASES
AUTHORS: Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Simo, Claude U. Konchie; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarem, Nuno; Tavares, Joana; Cordeiro da Silva, Anabela; Costi, Maria Paola; Tonelli, Michele;
PUBLISHED: 2024, SOURCE: ACS INFECTIOUS DISEASES
INDEXED IN: Scopus WOS
Scopus WOS3
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1 Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: WOS
WOS4
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1 Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
INDEXED IN: WOS
WOS5
TITLE: Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
AUTHORS: Carolina B Moraes; Gesa Witt; Maria Kuzikov; Bernhard Ellinper; Theodora Calogeropoulou; Kyriakos C Prousis; Stefano Mangani; Flavio Di Pisa; Giacomo Landi; Lucia Dello Lacono; Cecilia Pozzi; Lucio H Freitas Junior; Bruno dos Santos Pascoalino; Claudia P Bertolacini; Birte Behrens; Oliver Keminer; Jennifer Leu; Markus Wolf; Jeanette Reinshagen; Anabela Cordeiro da Silva ; ...More
PUBLISHED: 2019, SOURCE: SLAS DISCOVERY, VOLUME: 24, ISSUE: 3
AUTHORS: Carolina B Moraes; Gesa Witt; Maria Kuzikov; Bernhard Ellinper; Theodora Calogeropoulou; Kyriakos C Prousis; Stefano Mangani; Flavio Di Pisa; Giacomo Landi; Lucia Dello Lacono; Cecilia Pozzi; Lucio H Freitas Junior; Bruno dos Santos Pascoalino; Claudia P Bertolacini; Birte Behrens; Oliver Keminer; Jennifer Leu; Markus Wolf; Jeanette Reinshagen; Anabela Cordeiro da Silva ; ...More
PUBLISHED: 2019, SOURCE: SLAS DISCOVERY, VOLUME: 24, ISSUE: 3
6
TITLE: Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections Full Text
AUTHORS: Pasquale Linciano; Cecilia Pozzi; Lucia dello Iacono; Flavio di Pisa; Giacomo Landi; Alessio Bonucci; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Gesa Witt; Nuno Santarem; Catarina Baptista; Caio Franco; Carolina B Moraes; Wolfgang Mueller; Ulrike Wittig; Rosaria Luciani; Antony Sesenna; Antonio Quotadamo; Stefania Ferrari; ...More
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 8
AUTHORS: Pasquale Linciano; Cecilia Pozzi; Lucia dello Iacono; Flavio di Pisa; Giacomo Landi; Alessio Bonucci; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Gesa Witt; Nuno Santarem; Catarina Baptista; Caio Franco; Carolina B Moraes; Wolfgang Mueller; Ulrike Wittig; Rosaria Luciani; Antony Sesenna; Antonio Quotadamo; Stefania Ferrari; ...More
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 8
7
TITLE: Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors
AUTHORS: Giacomo Landi; Pasquale Linciano; Chiara Borsari; Claudia P Bertolacini; Carolina B Moraes; Anabela Cordeiro da Silva ; Sheraz Gul; Gesa Witt; Maria Kuzikov; Maria Paola Costi; Cecilia Pozzi; Stefano Mangani;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 7
AUTHORS: Giacomo Landi; Pasquale Linciano; Chiara Borsari; Claudia P Bertolacini; Carolina B Moraes; Anabela Cordeiro da Silva ; Sheraz Gul; Gesa Witt; Maria Kuzikov; Maria Paola Costi; Cecilia Pozzi; Stefano Mangani;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 7
8
TITLE: Chroman-4-One Derivatives Targeting Pteridine Reductase 1 and Showing Anti-Parasitic Activity Full Text
AUTHORS: Flavio Di Pisa; Giacomo Landi; Lucia Dello Iacono; Cecilia Pozzi; Chiara Borsari; Stefania Ferrari; Matteo Santucci; Nuno Santarem; Anabela Cordeiro da Silva ; Carolina B Moraes; Laura M Alcantara; Vanessa Fontana; Lucio H Freitas Junior; Sheraz Gul; Maria Kuzikov; Birte Behrens; Ina Poehner; Rebecca C Wade; Maria Paola Costi; Stefano Mangani;
PUBLISHED: 2017, SOURCE: MOLECULES, VOLUME: 22, ISSUE: 3
AUTHORS: Flavio Di Pisa; Giacomo Landi; Lucia Dello Iacono; Cecilia Pozzi; Chiara Borsari; Stefania Ferrari; Matteo Santucci; Nuno Santarem; Anabela Cordeiro da Silva ; Carolina B Moraes; Laura M Alcantara; Vanessa Fontana; Lucio H Freitas Junior; Sheraz Gul; Maria Kuzikov; Birte Behrens; Ina Poehner; Rebecca C Wade; Maria Paola Costi; Stefano Mangani;
PUBLISHED: 2017, SOURCE: MOLECULES, VOLUME: 22, ISSUE: 3
9
TITLE: Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit Trypanosoma brucei Pteridine Reductase in Support of Early-Stage Drug Discovery
AUTHORS: Linciano, P; Dawson, A; Pohner, I; Costa, DM; Sa, MS; Cordeiro da Silva, A ; Luciani, R; Gul, S; Witt, G; Ellinger, B; Kuzikov, M; Gribbon, P; Reinshagen, J; Wolf, M; Behrens, B; Hannaert, V; Michels, PAM; Nerini, E; Pozzi, C; di Pisa, F; ...More
PUBLISHED: 2017, SOURCE: ACS OMEGA, VOLUME: 2, ISSUE: 9
AUTHORS: Linciano, P; Dawson, A; Pohner, I; Costa, DM; Sa, MS; Cordeiro da Silva, A ; Luciani, R; Gul, S; Witt, G; Ellinger, B; Kuzikov, M; Gribbon, P; Reinshagen, J; Wolf, M; Behrens, B; Hannaert, V; Michels, PAM; Nerini, E; Pozzi, C; di Pisa, F; ...More
PUBLISHED: 2017, SOURCE: ACS OMEGA, VOLUME: 2, ISSUE: 9
10
TITLE: Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs Full Text
AUTHORS: Chiara Borsari; Rosaria Luciani; Cecilia Pozzi; Ina Poehner; Stefan Henrich; Matteo Trande; Anabela Cordeiro da Silva ; Nuno Santarem; Catarina Baptista; Annalisa Tait; Flavio Di Pisa; Lucia Dello Iacono; Giacomo Landi; Sheraz Gul; Markus Wolf; Maria Kuzikov; Bernhard Ellinger; Jeanette Reinshagen; Gesa Witt; Philip Gribbon; ...More
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
AUTHORS: Chiara Borsari; Rosaria Luciani; Cecilia Pozzi; Ina Poehner; Stefan Henrich; Matteo Trande; Anabela Cordeiro da Silva ; Nuno Santarem; Catarina Baptista; Annalisa Tait; Flavio Di Pisa; Lucia Dello Iacono; Giacomo Landi; Sheraz Gul; Markus Wolf; Maria Kuzikov; Bernhard Ellinger; Jeanette Reinshagen; Gesa Witt; Philip Gribbon; ...More
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
