M. S. Gadd
AuthID: R-00J-S90
1
TITLE: Group-Based Optimization of Potent and Cell-Active Inhibitors of the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase: Structure-Activity Relationships Leading to the Chemical Probe (2S,4R)-1-((S)-2-(1-Cyanocyclopropanecarboxamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide (VH298) Full Text
AUTHORS: Soares, P ; Gadd, MS; Frost, J; Galdeano, C; Ellis, L; Epemolu, O; Rocha, S; Read, KD; Ciulli, A;
PUBLISHED: 2018, SOURCE: Journal of Medicinal Chemistry, VOLUME: 61, ISSUE: 2
AUTHORS: Soares, P ; Gadd, MS; Frost, J; Galdeano, C; Ellis, L; Epemolu, O; Rocha, S; Read, KD; Ciulli, A;
PUBLISHED: 2018, SOURCE: Journal of Medicinal Chemistry, VOLUME: 61, ISSUE: 2
