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TITLE: Oxetane Grafts Installed Site‐Selectively on Native Disulfides to Enhance Protein Stability and Activity In Vivo
AUTHORS: Nuria Martínez‐Sáez; Shuang Sun; Davide Oldrini; Pietro Sormanni; Omar Boutureira; Filippo Carboni; Ismael Compañón; Michael J Deery; Michele Vendruscolo; Francisco Corzana; Roberto Adamo; Gonçalo J L Bernardes;
PUBLISHED: 2017, SOURCE: Angewandte Chemie International Edition, VOLUME: 56, ISSUE: 47
INDEXED IN: CrossRef: 39
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62
TITLE: Oxetane Grafts Installed Site‐Selectively on Native Disulfides to Enhance Protein Stability and Activity In Vivo
AUTHORS: Nuria Martínez‐Sáez; Shuang Sun; Davide Oldrini; Pietro Sormanni; Omar Boutureira; Filippo Carboni; Ismael Compañón; Michael J Deery; Michele Vendruscolo; Francisco Corzana; Roberto Adamo; Gonçalo J L Bernardes;
PUBLISHED: 2017, SOURCE: Angewandte Chemie, VOLUME: 129, ISSUE: 47
INDEXED IN: CrossRef: 10
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63
TITLE: Precise Probing of Residue Roles by Post-Translational β,γ-C,N Aza-Michael Mutagenesis in Enzyme Active Sites
AUTHORS: Jitka Dadová; Kuan-Jung Wu; Patrick G Isenegger; James C Errey; Gonçalo J L Bernardes; Justin M Chalker; Lluís Raich; Carme Rovira; Benjamin G Davis;
PUBLISHED: 2017, SOURCE: ACS Central Science, VOLUME: 3, ISSUE: 11
INDEXED IN: CrossRef: 33
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64
TITLE: Iminoboronates are efficient intermediates for selective, rapid and reversible N-terminal cysteine functionalisation
AUTHORS: Faustino, H; Silva, MJSA; Veiros, LF; Bernardes, GJL; Gois, PMP;
PUBLISHED: 2016, SOURCE: CHEMICAL SCIENCE, VOLUME: 7, ISSUE: 8
INDEXED IN: Scopus WOS CrossRef
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65
TITLE: Tn Antigen Mimics Based on sp2-Iminosugars with Affinity for an anti-MUC1 Antibody  Full Text
AUTHORS: Fernández, EMS; Navo, CD; Martínez Sáez, N; Gonçalves Pereira, R; Somovilla, VJ; Avenoza, A; Busto, JH; Bernardes, GJL; Jiménez Osés, G; Corzana, F; Fernández, JMG; Mellet, CO; Peregrina, JM;
PUBLISHED: 2016, SOURCE: Organic Letters, VOLUME: 18, ISSUE: 15
INDEXED IN: Scopus CrossRef
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66
TITLE: Stoichiometric and irreversible cysteine-selective protein modification using carbonylacrylic reagents
AUTHORS: Bernardim, B; Cal, PMSD; Matos, MJ ; Oliveira, BL; Martinez Saez, N; Albuquerque, IS; Perkins, E; Corzana, F; Burtoloso, ACB; Jimenez Oses, G; Bernardes, GJL;
PUBLISHED: 2016, SOURCE: NATURE COMMUNICATIONS, VOLUME: 7, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 137
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67
TITLE: Natural product modulators of transient receptor potential (TRP) channels as potential anti-cancer agents
AUTHORS: Rodrigues, T; Sieglitz, F; Bernardes, GJL;
PUBLISHED: 2016, SOURCE: CHEMICAL SOCIETY REVIEWS, VOLUME: 45, ISSUE: 22
INDEXED IN: Scopus WOS CrossRef: 57
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68
TITLE: Posttranslational mutagenesis: A chemical strategy for exploring protein side-chain diversity
AUTHORS: Wright, TH; Bower, BJ; Chalker, JM; Bernardes, GJL; Wiewiora, R; Ng, WL; Raj, R; Faulkner, S; Vallee, MRJ; Phanumartwiwath, A; Coleman, OD; Thezenas, ML; Khan, M; Galan, SRG; Lercher, L; Schombs, MW; Gerstberger, S; Palm Espling, ME; Baldwin, AJ; Kessler, BM; Claridge, TDW; Mohammed, S; Davis, BG; ...More
PUBLISHED: 2016, SOURCE: SCIENCE, VOLUME: 354, ISSUE: 6312
INDEXED IN: Scopus WOS CrossRef: 247
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69
TITLE: A Minimal, Unstrained S-Allyl Handle for Pre-Targeting Diels-Alder Bioorthogonal Labeling in Live Cells
AUTHORS: Oliveira, BL; Guo, ZJ; Boutureira, O; Guerreiro, A; Jimenez Oses, G; Bernardes, GJL;
PUBLISHED: 2016, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 55, ISSUE: 47
INDEXED IN: WOS CrossRef: 27
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70
TITLE: Construction of homogeneous antibody-drug conjugates using site-selective protein chemistry
AUTHORS: Akkapeddi, P; Azizi, SA; Freedy, AM; Cal, PMSD; Gois, PMP; Bernardes, GJL;
PUBLISHED: 2016, SOURCE: CHEMICAL SCIENCE, VOLUME: 7, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 130
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