21
TITLE: Structure-Activity Relationship Studies and Plasmodium Life Cycle Profiling Identifies Pan-Active N-Aryl-3-trifluoromethyl Pyrido[1,2-a]benzimidazoles Which Are Efficacious in an in Vivo Mouse Model of Malaria  Full Text
AUTHORS: Godfrey Mayoka; Mathew Njoroge; John Okombo; Liezl Gibhard; Margarida Sanches Vaz; Diana Fontinha; Lyn Marie Birkholtz; Janette Reader; Mariette van der Watt; Theresa L Coetzer; Sonja Lauterbach; Alisje Churchyard; Belinda Bezuidenhout; Timothy J Egan; Clive Yeates; Sergio Wittlin; Miguel Prudencio ; Kelly Chibale;
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
22
TITLE: Synthesis and antiplasmodial evaluation of novel mefloquine-based fumardiamides  Full Text
AUTHORS: Maja Beus; Diana Fontinha; Jana Held; Zrinka Rajic; Miguel Prudencio ; Branka Zorc;
PUBLISHED: 2019, SOURCE: ACTA PHARMACEUTICA, VOLUME: 69, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
24
TITLE: Primaquine homodimers as potential antiplasmodial and anticancer agents  Full Text
AUTHORS: Kristina Pavic; Barbara Rubinic; Zrinka Rajic; Diana Fontinha; Miguel Prudencio ; Lidija Uzelac; Marijeta Kralj; Jana Held; Branka Zorc;
PUBLISHED: 2019, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, VOLUME: 29, ISSUE: 19
INDEXED IN: Scopus WOS
25
TITLE: Primaquine and Chloroquine Fumardiamides as Promising Antiplasmodial Agents  Full Text
AUTHORS: Maja Beus; Diana Fontinha; Jana Held; Zrinka Rajic; Lidija Uzelac; Marijeta Kralj; Miguel Prudencio ; Branka Zorc;
PUBLISHED: 2019, SOURCE: MOLECULES, VOLUME: 24, ISSUE: 15
INDEXED IN: Scopus WOS CrossRef: 1
26
TITLE: Flexible 3D Cell-Based Platforms for the Discovery and Profiling of Novel Drugs Targeting Plasmodium Hepatic Infection
AUTHORS: Francisca Arez; Sofia P Rebelo; Diana Fontinha; Daniel Simao; Tatiana R Martins; Marta Machado; Christoph Fischli; Claude Oeuvray; Lassina Badolo; Manuel J T Carrondo; Matthias Rottmann; Thomas Spangenberg; Catarina Brito; Beatrice Greco; Miguel Prudencio; Paula M Alves;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef: 1
27
TITLE: Primaquine homodimers as potential antiplasmodial and anticancer agents  Full Text
AUTHORS: Kristina Pavić; Barbara Rubinić; Zrinka Rajić; Diana Fontinha; Miguel Prudêncio; Lidija Uzelac; Marijeta Kralj; Jana Held; Branka Zorc;
PUBLISHED: 2019, SOURCE: Bioorganic & Medicinal Chemistry Letters, VOLUME: 29, ISSUE: 19
INDEXED IN: CrossRef
28
TITLE: Primaquine hybrids as promising antimycobacterial and antimalarial agents  Full Text
AUTHORS: Kristina Pavic; Ivana Perkovic; Sarka Pospisilova; Marta Machado; Diana Fontinha; Miguel Prudencio ; Josef Jampilek; Aidan Coffey; Lorraine Endersen; Hrvoje Rimac; Branka Zorc;
PUBLISHED: 2018, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 143
INDEXED IN: Scopus WOS
29
TITLE: SAHAquines, Novel Hybrids Based on SAHA and Primaquine Motifs, as Potential Cytostatic and Antiplasmodial Agents  Full Text
AUTHORS: Maja Beus; Zrinka Rajic; Dusica Maysinger; Zvonimir Mlinaric; Maja Antunovic; Inga Marijanovic; Diana Fontinha; Miguel Prudencio ; Jana Held; Sureyya Olgen; Branka Zorc;
PUBLISHED: 2018, SOURCE: CHEMISTRYOPEN, VOLUME: 7, ISSUE: 8
INDEXED IN: Scopus WOS CrossRef
30
TITLE: A HUMAN 3D CELL-BASED PLATFORM FOR DRUG DISCOVERY TARGETING PLASMODIUM HEPATIC INFECTION
AUTHORS: Sofia Rebelo; Francisca Arez; Diana Fontinha; Daniel Simao; Marta Machado; Tatiana Martins; Manuel Carrondo; Thomas Spangenberg; Catarina Brito; Beatrice Greco; Miguel Prudencio; Paula Alves;
PUBLISHED: 2018, SOURCE: 67th Annual Meeting of the American-Society-of-Tropical-Medicine-and-Hygiene (ASTHM) in AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, VOLUME: 99, ISSUE: 4
INDEXED IN: WOS
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