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TITLE: Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign  Full Text
AUTHORS: Pasquale Linciano; Gregorio Cullia; Chiara Borsari; Matteo Santucci; Stefania Ferrari; Gesa Witt; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Nuno Santarem; Anabela Cordeiro da Silva ; Paola Conti; Maria Laura Bolognesi; Marinella Roberti; Federica Prati; Francesca Bartoccini; Michele Retini; Giovanni Piersanti; Andrea Cavalli; Luca Goldoni; Sine Mandrup Bertozzi; Fabio Bertozzi; Enzo Brambilla; Vincenzo Rizzo; Daniele Piomelli; Andrea Pinto; Tiziano Bandiera; Maria Paola Costi; ...More
PUBLISHED: 2020, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 189
INDEXED IN: Scopus WOS CrossRef
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TITLE: Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity  Full Text
AUTHORS: Thomas C Eadsforth; Andrea Pinto; Rosaria Luciani; Lucia Tamborini; Gregorio Cullia; Carlo De Micheli; Luciana Marinelli; Sandro Cosconati; Ettore Novellino; Leonardo Lo Presti; Anabela Cordeiro da Silva ; Paola Conti; William N Hunter; Maria P Costi;
PUBLISHED: 2015, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 58, ISSUE: 20
INDEXED IN: Scopus WOS CrossRef